| Simcere Zaiming, Inc. | Former 10% Owner | 30,000Common Stock | — | Sell | |
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| ADAR1 Capital Management, LLC | 10% Owner | 36,303Common Stock | — | Buy | |
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| ADAR1 Capital Management, LLC | 10% Owner | 272,850Common Stock | — | Buy | |
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| ADAR1 Capital Management, LLC | 10% Owner | 3,410Common Stock | — | Buy | |
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| ADAR1 Capital Management, LLC | 10% Owner | 6,400Common Stock | — | Buy | |
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| ADAR1 Capital Management, LLC | 10% Owner | 7,798Common Stock | — | Buy | |
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| Webster Stephen W | Director | 2,340Stock Option (Right to Buy) | — | Grant / award | |
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| KABAKOFF DAVID S | Director | 3,510Stock Option (Right to Buy) | — | Grant / award | |
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| Jones Elaine V | Director | 2,340Stock Option (Right to Buy) | — | Grant / award | |
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| Houston John G | Director | 2,340Stock Option (Right to Buy) | — | Grant / award | |
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